Half-Life Reference Chart

A static, at-a-glance reference for approximate half-lives of common peptides and the dosing frequency each implies. Half-life is roughly the time for blood levels to fall by half; a short half-life usually means more frequent dosing, a long one allows less frequent dosing. For the concepts behind this table, see Half-Life & Pharmacokinetics.

Read this first

These values are approximate and many are drawn from limited or animal data. Where human pharmacokinetics are poorly characterized, the cell says “approx” or “not well established.” Half-life is only one input into dosing — receptor kinetics, the duration of the downstream effect (e.g. a GH pulse), and clinical context all matter. This is educational, not a dosing recommendation.

Reference table

PeptideApprox half-lifeTypical dosing frequencyNotes
BPC-157~minutes (approx; animal data)1–2× dailyHuman PK not well established; short systemic half-life but locally acting; route-dependent
TB-500Not well established (approx hours, route-dependent)~1–2× weeklyFull Tβ4 reported ~hours; community protocols use a weekly “loading/maintenance” pattern
CJC-1295 without DAC (Mod GRF 1-29)~30 minutes (approx)Multiple times dailyVery short; designed to mimic a single GH pulse; often paired with Ipamorelin
CJC-1295 with DAC~6–8 days~1–2× weeklyDAC binds albumin for a slow-release depot; sustained (less pulsatile) GH/IGF-1 rise
Ipamorelin~2 hours1–3× dailyGH peak ~0.67 h after dosing then rapid decline; injectable (destroyed in gut)
MK-677~24 hoursOnce dailyOrally active non-peptide ghrelin mimetic; sustained 24-h GH/IGF-1 elevation
Sermorelin~10–20 minutesOnce daily (usually bedtime)Very short; GHRH analog; often timed to nocturnal GH pulse
Tesamorelin~11 minutes (SC, healthy subjects)Once dailyShort half-life but once-daily per FDA labeling (Egrifta)
Semaglutide~7 days (~160 h)Once weeklyGLP-1 analog; fatty-diacid albumin binding enables weekly dosing
Tirzepatide~5 daysOnce weeklyDual GIP/GLP-1 agonist; albumin-binding chain enables weekly dosing
Retatrutide~6 daysOnce weeklyInvestigational triple GIP/GLP-1/glucagon agonist; dose-proportional PK
PT-141~2.7 h (range ~1.9–4.0 h)On demandShort half-life fits its as-needed use pattern
SS-31~ a few hours (SC; approx)Once dailyMitochondria-targeting tetrapeptide (elamipretide); indication-dependent
Thymosin Alpha-1~2 hours~2× weeklyApproved-abroad regimen (thymalfasin) is 1.6 mg twice weekly
Kisspeptin~4 min (Kp-10); Kp-54 ~28 minInfusion (trials)Very short; trials use IV infusion or the longer Kp-54 fragment
EpitalonVery short (~minutes; approx)Daily in short coursesRapidly hydrolyzed; human PK not well characterized; typically dosed in 10–20 day courses

How to read it

  • Short half-life (minutes to a few hours) — e.g. Sermorelin, Tesamorelin, no-DAC CJC-1295, Ipamorelin, PT-141. These clear quickly, so they are dosed daily, several times daily, or on demand. A short half-life is often intentional for GH secretagogues, which aim to mimic the body’s natural brief pulses rather than a constant elevation.
  • Long half-life (days) — e.g. CJC-1295 with DAC, Semaglutide, Tirzepatide, Retatrutide. Albumin binding (or, for the GLP-1 class, a fatty-acid chain) extends these to days, enabling once-weekly dosing.
  • Poorly characterized — e.g. BPC-157, TB-500, Epitalon. Systemic half-life is uncertain in humans; dosing frequency in these cases comes from community/empirical practice, not robust PK studies.

For side-by-side comparisons across more attributes, see Comparison Tables and Stacks & Comparisons.


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Educational information only — not medical advice. See Disclaimer.